STO-609 是选择性和细胞可渗透的 CaM-KK 抑制剂,对重组 CaM-KKα 和 CaM-KKβ 的Ki值分别为 80 和 15 ng/mL。STO-609 抑制 Hela 细胞溶解物中的 AMP 活化蛋白激酶激酶 (AMPKK) 活性,IC50 值为 ~0.02 g/ml。
Cas No. | 52029-86-4 | SDF | |
别名 | N/A | ||
化学名 | N/A | ||
Canonical SMILES | O=C(C1=C2C3=C(C4=NC5=CC=CC=C5N4C(C3=CC=C2)=O)C=C1)O | ||
分子式 | C19H10N2O3 | 分子量 | 314.29 |
溶解度 | DMSO: 5.6 mg/mL (17.82 mM and warming); Water: < 0.1 mg/mL (insoluble) | 储存条件 | Store at -20°C |
General tips | For obtaining a higher solubility , please warm the tube at 37 ℃ and shake it in the ultrasonic bath for a while. | ||
Shipping Condition |
Evaluation sample solution : ship with blue ice All other available size: ship with RT , or blue ice upon request |