PF-CBP1 HCl is a highly selective inhibitor of the bromodomain of CREB-binding protein(CREBBP). It inhibits CREBBP (IC50: 125 nM) and p300 bromodomains (IC50: 363 nM).
| 常用名 | PF-CBP1 hydrochloride | 英文名 | PF-CBP1 hydrochloride |
|---|---|---|---|
| CAS号 | 1962928-21-7 | 分子量 | 488.621 |
| 密度 | 1.2±0.1 g/cm3 | 沸点 | 673.5±55.0 °C at 760 mmHg |
| 分子式 | C29H36N4O3 | 熔点 | N/A |
| MSDS | N/A | 闪点 | 361.1±31.5 °C |